E-Dissertationen: Search
Now showing items 1-4 of 4
Elucidating agonist-induced signaling patterns of human G protein-coupled receptor GPR17 and uncovering pranlukast as a biased mixed agonist-antagonist at GPR17
(2011-11-15)
The progress of human genome sequencing has revealed the existence of several hundred orphan G protein-coupled receptors (GPCRs), whose endogenous ligands are not yet identified, thus their deorphanization and characterization ...
A2B-Adenosin-Rezeptor-Homo- und Heterodimere: Biolumineszenz-Resonanz-Energie-Transfer-Studien und pharmakologische Charakterisierung
(2012-12-12)
Die Adenosin-Rezeptoren, welche zur Superfamilie der G-Protein-gekoppelten Rezeptoren (GPCR) gehören, werden in die vier Subtypen, A1, A2A, A2B und A3 unterteilt. Aufgrund der ...
EBI2 is a negative modulator of adipose tissue activity
(2020-08-17)
Weight-related diseases are common and often fatal conditions characterized by an imbalance between energy intake and energy expenditure. Obesity and weight gain related diseases such as type 2-diabetes have reached in the ...
Medizinische Chemie und molekulare Pharmakologie G-Protein-gekoppelter Purin- und verwandter Waisen-Rezeptoren
(2014-06-17)
G-Protein-gekoppelte Rezeptoren gehören zu den wichtigsten pharmakologischen Zielstrukturen. Für einige dieser Rezeptoren wurden purinerge Verbindungen (Adenin-Nucleotide, Adenosin und Adenin) als endogene Agonisten ...